Warheads
Selected indexed studies
- Electrophilic warheads in covalent drug discovery: an overview. (Expert Opin Drug Discov, 2022) [PMID:35129005]
- Emerging and Re-emerging Warheads for Targeted Covalent Inhibitors: An Update. (J Med Chem, 2024) [PMID:38711345]
- Covalent Warheads Targeting Cysteine Residue: The Promising Approach in Drug Development. (Molecules, 2022) [PMID:36431829]
_Worker-drafted node — pending editorial review._
Connections
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Sources
- Electrophilic warheads in covalent drug discovery: an overview. (2022) pubmed
- Emerging and Re-emerging Warheads for Targeted Covalent Inhibitors: An Update. (2024) pubmed
- Covalent Warheads Targeting Cysteine Residue: The Promising Approach in Drug Development. (2022) pubmed
- Systematic Exploration of Privileged Warheads for Covalent Kinase Drug Discovery. (2022) pubmed
- The expanding repertoire of covalent warheads for drug discovery. (2023) pubmed
- Covalent drug discovery using sulfur(VI) fluoride exchange warheads. (2023) pubmed
- Recent progress in covalent warheads for in vivo targeting of endogenous proteins. (2021) pubmed
- Recent advances in the design of small molecular drugs with acrylamides covalent warheads. (2024) pubmed
- Emerging and Re-Emerging Warheads for Targeted Covalent Inhibitors: Applications in Medicinal Chemistry and Chemical Biology. (2019) pubmed
- Bicyclobutanes: from curiosities to versatile reagents and covalent warheads. (2022) pubmed